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2016 Vol. 24, No. 4
Published: 20 April 2016

 
277 Synthesis and Biological Evaluation of Novel PARP-1 Inhibitors with Indazole Skeleton
LONG Wei, QIU Wen-ge, HU Yun-yan, SONG Li-yun, LI Hai-jun, HE Hong
DOI: 10.15952/j.cnki.cjsc.1005-1511.2016.04.16016
2016 Vol. 24 (4): 277-282 [Abstract] ( 375 ) HTML (1 KB)  PDF (1097 KB)  ( 324 )
283 Synthesis and Antitumor Activities of Novel N6-Piperazine Substituted Adenosine Analogues
ZHOU Gao-hui, LUO Ming-ming, ZHANG Yang,YU Xiao-qin, TAO Li-ming, XU Wen-ping
DOI: 10.15952/j.cnki.cjsc.1005-1511.2016.04.15151
2016 Vol. 24 (4): 283-287 [Abstract] ( 300 ) HTML (1 KB)  PDF (797 KB)  ( 268 )
288 Synthesis and Biologial Activities of Novel Magnolol -2-Azomethine Derivatives
MEI Fan, ZHAI Ting, ZHENG Nian, LI Yan, CHEN Yong, LOU Zhao-wen
DOI: 10.15952/j.cnki.cjsc.1005-1511.2016.04.15145
2016 Vol. 24 (4): 288-292 [Abstract] ( 356 ) HTML (1 KB)  PDF (653 KB)  ( 308 )
293 Synthesis and Antitumor Activities of Novel Indazole Derivatives
ZHOU Yun-peng, HE Chang, SONG Duan-zheng, CHEN Ye, LIU Ju, ZHANG Qiu-shi, WANG Yang
DOI: 10.15952/j.cnki.cjsc.1005-1511.2016.04.16019
2016 Vol. 24 (4): 293-296 [Abstract] ( 401 ) HTML (1 KB)  PDF (588 KB)  ( 284 )
297 Synthesis and Anti-platelet Aggregation Activities of Novel Thienopyridine Derivatives
FAN Meng-lin, JIANG Xi-ming, LIU Ying, LIU Deng-ke, WANG Ping-bao
DOI: 10.15952/j.cnki.cjsc.1005-1511.2016.04.15393
2016 Vol. 24 (4): 297-301 [Abstract] ( 342 ) HTML (1 KB)  PDF (643 KB)  ( 313 )
302 Preparation of Three-dimensional Porous Reduced Graphene Oxide Aerogel and Its Application in Lithium-ion Batteries
DENG Xiao-mei, WEN Hao, ZHANG Chu-hong, DENG Jian-guo, GAO Li-zhen
DOI: 10.15952/j.cnki.cjsc.1005-1511.2016.04.15073
2016 Vol. 24 (4): 302-307 [Abstract] ( 501 ) HTML (1 KB)  PDF (1673 KB)  ( 879 )
308 Synthesis of Novel Choline Derivatives and Their in vitro Antimalarial Activities
WANG Fang, ZHAO Qing, CHEN Hui-fang, ZHANG Shu-qiu
DOI: 10.15952/j.cnki.cjsc.1005-1511.2016.04.15415
2016 Vol. 24 (4): 308-311 [Abstract] ( 235 ) HTML (1 KB)  PDF (582 KB)  ( 281 )
312 Synthesis  of A Novel Mono-hydroxyl Chloro-corrole and Its Photocleavage of DNA
SHI Lei, YANG Wen-cong, ZENG Shu-ying,MO Ting-ting, WANG Hua-hua, LIU Hai-yang
DOI: 10.15952/j.cnki.cjsc.1005-1511.2016.04.15408
2016 Vol. 24 (4): 312-315 [Abstract] ( 316 ) HTML (1 KB)  PDF (695 KB)  ( 256 )
316 Synthesis of Novel Potassium(3-fluoro-2-amino-substituted pyridin-4-yltrifluoroborates)
TENG Ming-gang, ZHAO Chun-shen, DUAN Lian, CHAI Hui-fang
DOI: 10.15952/j.cnki.cjsc.1005-1511.2016.04.15146
2016 Vol. 24 (4): 316-320 [Abstract] ( 333 ) HTML (1 KB)  PDF (583 KB)  ( 310 )
321 Synthesis of Xanthenes Catalyzed by Ionic Liquid 1-Ethyl-3-(4-sulfobutyl)-1H-imidazol-3-ium -p-Toluenesulfonate
TIAN Xiao-yue, ZHANG Yong-hong, SUN Ya-dong, WANG Duo-zhi, LIU Chen-jiang
DOI: 10.15952/j.cnki.cjsc.1005-1511.2016.04.15153
2016 Vol. 24 (4): 321-325 [Abstract] ( 303 ) HTML (1 KB)  PDF (654 KB)  ( 462 )
326 A New Synthetic Method of α-Sulfo-β-amino Acid Esters
HU Xiao-yan, HU Fang-zhi, YUAN Wei-cheng, ZHANG Xiao-mei
DOI: 10.15952/j.cnki.cjsc.1005-1511.2016.04.15164
2016 Vol. 24 (4): 326-329 [Abstract] ( 317 ) HTML (1 KB)  PDF (332 KB)  ( 280 )
330 Organocatalytic Asymmetric Michael Addition of Barbituric Acid to β-Nitroalkenes
GUI Yong-yuan, LIU Kang-qiong, WANG Xiao, TIAN Fang, PENG Lin, WANG Li-xin
DOI: 10.15952/j.cnki.cjsc.1005-1511.2016.04.15183
2016 Vol. 24 (4): 330-332 [Abstract] ( 343 ) HTML (1 KB)  PDF (535 KB)  ( 296 )
333 Poly(p-dioxanone-co-Nε-carbobenzoxy-L-lysine):Synthesis and Mechanism of Copolymerization
WANG Bing, DONG Jun, CHEN Dong-liang, XIONG Cheng-dong
DOI: 10.15952/j.cnki.cjsc.1005-1511.2016.04.15149
2016 Vol. 24 (4): 333-337 [Abstract] ( 271 ) HTML (1 KB)  PDF (1629 KB)  ( 295 )
338 Synthesis and Photoisomerization Behavior of Azobenzene Compounds Containing Various Groups
LIU Jia, TIAN Jin-tao
DOI: 10.15952/j.cnki.cjsc.1005-1511.2016.04.15094
2016 Vol. 24 (4): 338-341 [Abstract] ( 516 ) HTML (1 KB)  PDF (1119 KB)  ( 608 )
342 Synthesis of Novel Sulfinyl-NH-olefine Ligands and Their Application in Transfer Hydrogenation Reaction
LIN Zhe-chao, TANG Lei, HUANG Qing-fei, WANG Qi-wei, DENG Jin-gen
DOI: 10.15952/j.cnki.cjsc.1005-1511.2016.04.15128
2016 Vol. 24 (4): 342-346 [Abstract] ( 289 ) HTML (1 KB)  PDF (487 KB)  ( 337 )
346 Synthesis and Crystal Structure of 2-(N-cyclohexylamine)-6-trifluoromethoxy-benzothiazole
WU Xiang-long, LIU Liu, LI You-jia, LUO Jie,GAI Dong-wei, MA Jing-chuan, MEI Qi-bing
DOI: 10.15952/j.cnki.cjsc.1005-1511.2016.04.15404
2016 Vol. 24 (4): 346-349 [Abstract] ( 383 ) HTML (1 KB)  PDF (890 KB)  ( 367 )
350 Asymmetric Hydroxylation of 1,2,3,4- Tetrahydroquinoline by Hydroxylase-catalyzed Hydroxylation in Two-phase Reaction System
LI Ke, YANG Min, CUI Bao-dong, CHEN Yong-zheng
DOI: 10.15952/j.cnki.cjsc.1005-1511.2016.04.16010
2016 Vol. 24 (4): 350-354 [Abstract] ( 333 ) HTML (1 KB)  PDF (628 KB)  ( 323 )
355 Synthesis of (3S,4S)-4-amino-3-hydroxy-5-phenylpentanoic  Acid Derivatives Catalyzed by D-proline
BAO Ke-ting, ZHANG Wei, LI Ying-xia, HU Chun
DOI: 10.15952/j.cnki.cjsc.1005-1511.2016.04.16006
2016 Vol. 24 (4): 355-358 [Abstract] ( 339 ) HTML (1 KB)  PDF (523 KB)  ( 391 )
359 A Novel Synthetic Method for Ginkgolic Acid
ZHAO Jian-yang, WANG Ting, LIU Qing-qing,ZHU Jin, HUANG Qing-fei, WANG Qi-wei
DOI: 10.15952/j.cnki.cjsc.1005-1511.2016.04.15395
2016 Vol. 24 (4): 359-361 [Abstract] ( 324 ) HTML (1 KB)  PDF (496 KB)  ( 327 )
362 Research Process on Preparation ofNovel Macromolecular by ATRP/CuAAC Technique
WEI Ke-yao, JI Hu, WU Qi, ZHAO Xin,DUAN Ran, LEI Liang-cai, LI Hai-ying
DOI: 10.15952/j.cnki.cjsc.1005-1511.2016.04.16003
2016 Vol. 24 (4): 362-368 [Abstract] ( 369 ) HTML (1 KB)  PDF (1735 KB)  ( 388 )
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